An advanced automated patch clamp protocol design to investigate drug - ion channel binding dynamics.
P. Lukacs, K. Pesti, M. C. Foldi, K. Zboray, A. V. Toth, G. Papp, A. Mike
This study introduces an automated patch-clamp protocol to assess drug-sodium channel binding dynamics, revealing complex on- and off-kinetics across multiple time scales.
bioRxiv · Jul 5, 2021Pharmacology & Toxicology