Drug design and repurposing with a sequence-to-drug paradigm
Lifan Chen, Zisheng Fan, Jie Chang, Ruirui Yang, Hao Guo, Yinghui Zhang, Tianbiao Yang, Chenmao Zhou, Zhengyang Chen, Chen Zheng, Xinyue Hao, Keke Zhang, Rongrong Cui, Yiluan Ding, Naixia Zhang, , Mingyue Zheng
This paper introduces a sequence-to-drug paradigm using TransformerCPI2.0 to discover drug-like molecules from protein sequences and validates its effectiveness for three targets.
bioRxiv · Mar 26, 2022 · PreprintMolecular Biology