The 11β-hydroxysteroid dehydrogenase type 1 inhibitor SPI-62 prevents morbidity in a mouse model of Cushing's syndrome
Xingyu Pan, Qiongqiong Hou, Jing Su, Jiahui Xu, Min Li, Jiawen Li, Xuerou Shi, Caleb Schmicker, Tobias Magers, William M Bracken, David A. Katz
SPI-62, an HSD-1 inhibitor, reduces GC-induced morbidity in a mouse Cushing's syndrome model by improving insulin sensitivity, reducing adiposity, and preventing skeletal myopathy.
bioRxiv · May 27, 2024 · PreprintPharmacology & Toxicology