Partial agonists and heteromeric Kainate receptor desensitization
Nami Tajima, Guadalupe Segura-Covarrubias, Ashlee M'Kay Hoffman, Changping Zhou
This study investigates how partial agonists affect desensitization in KARs, showing that agonist residence time and LBD closure are more critical than subunit composition in heteromeric receptors.
bioRxiv · Nov 3, 2026 · PreprintPhysiology