Activation of ARTD2/PARP2 by DNA damage induces conformational changes relieving enzyme autoinhibition
E. Obaji, M. M. Maksimainen, A. Galera-Prat, L. Lehtio
The paper describes how DNA damage activates ARTD2/PARP2 through conformational changes that relieve autoinhibition and enable catalytic activity.
bioRxiv · Nov 24, 2020Biochemistry