Chemoproteomic Characterization of GPX4 Covalent Ligands and Targeted Degradation
Vilas D. Kadam, Guangcan Bai, Chen Mozes, Hanling Guo, Zhouyiyuan Xue, Qi Miao, Jian Wang, Minhua Li, Feng Li, Daisuke Nakada, Zhi Tan, Xiaoyu Zhang, Mingxing Teng
The paper characterizes a covalent GPX4 inhibitor and develops degraders, expanding tools for GPX4 targeting.
bioRxiv · May 3, 2026 · PreprintCancer Biology