Radiosynthesis and Evaluation of Novel Cholesterol 24-Hydroxylase Positron Emission Tomography Tracers
Yinlong Li, Haofeng Shi, Zhendong Song, Taoqian Zhao, Yanwei Jiang, Danielle E. Hoyle, Jiahui Chen, Xin Zhou, Qilong Hu, Xiaoyan Li, Lingxin Meng, Ruihu Song, Zhenkun Sun, Ahmed Haider, Hongjie Yuan, Steven H. Liang
The paper designs and evaluates novel PET tracers for CYP46A1 by modifying cyclopropyl groups, showing high affinity and suitable radiosynthesis.
bioRxiv · Jan 27, 2026 · PreprintPharmacology & Toxicology