Bisphenol A derivatives act as novel coactivator binding inhibitors for estrogen receptor β
M. Iwamoto, T. Masuya, M. Hosose, K. Tagawa, T. Ishibashi, E. Yoshihara, M. Downes, R. M. Evans, A. Matsushima
This study identifies bisphenol A derivatives as novel coactivator binding inhibitors for estrogen receptor β, showing dual agonist/antagonist activities and a new ligand interaction site.
bioRxiv · May 10, 2021Biochemistry