Direct Small Molecule Activation of Mitofusins
Emmanouil Zacharioudakis, Nikolaos Biris, Thomas P. Garner, Yun Chen, Ryan Pekson, Rimpy Dhingra, Gaetano Santulli, Lorrie A. Kirshenbaum, Richard N. Kitsis, Evripidis Gavathiotis
This study identifies MASM7 as a direct activator of mitofusin 2, promoting mitochondrial fusion through conformational changes.
bioRxiv · Apr 17, 2018 · PreprintBiochemistry