Identification of 2-amino benzothiazoles with bactericidal activity against Mycobacterium tuberculosis
S. A. Bonnett, J.-A. Jee, S. Chettiar, Y. Ovechkina, A. Korkegian, E. Greve, J. Odingo, T. Parish
The paper identifies 2-amino benzothiazoles with bactericidal activity against Mycobacterium tuberculosis, showing improved potency and reduced cytotoxicity but poor metabolic stability.
bioRxiv · Sep 23, 2022 · PreprintMicrobiology