A Specific Non-Bisphosphonate Inhibitor Of The Bifunctional Farnesyl/Geranylgeranyl Diphosphate Synthase In Malaria Parasites
J. E. Gisselberg, Z. Herrera, L. Orchard, M. Llinas, E. Yeh
This paper identifies MMV019313 as a specific non-bisphosphonate inhibitor of PfFPPS/GGPPS in malaria parasites, showing superior properties and selectivity over bisphosphonates.
bioRxiv · Jul 21, 2017Microbiology