MicrobiologybioRxiv
A Specific Non-Bisphosphonate Inhibitor Of The Bifunctional Farnesyl/Geranylgeranyl Diphosphate Synthase In Malaria Parasites
J. E. Gisselberg, Z. Herrera, L. Orchard…·E. Yeh
This paper identifies MMV019313 as a specific non-bisphosphonate inhibitor of PfFPPS/GGPPS in malaria parasites, showing superior properties and selectivity over bisphosphonates.
DOI 10.1016/j.chembiol.2017.11.010