Pharmacology & ToxicologybioRxiv
Non-blocking modulation contributes to sodium channel inhibition by a covalently attached photoreactive riluzole analog
P. Lukacs, M. C. Foldi, L. Valanszki…·A. Mike
This study shows that non-blocking modulation of sodium channels is possible using a covalently attached photoreactive riluzole analog, suggesting new avenues for drug development.
DOI 10.1038/s41598-018-26444-y