Molecular insights into intrinsic transducer-coupling bias in the CXCR4-CXCR7 system
P. Sarma, H.-J. Yoon, C. M. Carino, D. S., R. Banerjee, Y. Yun, J. Ji, K. Min, S. Pandey, H. Dwivedi-Agnihotri, X. Rui, Y. Cao, K. Kawakami, Y.-C. Chen, P. Kumari, , A. K. Shukla
This study characterizes the biased agonism of CXCR4 and CXCR7, revealing differences in G-protein coupling, β-arrestin recruitment, and ERK1/2 activation.
bioRxiv · Jun 6, 2022Biochemistry