Directed biosynthesis of fluorinated polyketides
A. Rittner, M. Joppe, J. J. Schmidt, L. M. Mayer, E. Heid, D. H. Sherman, M. Grininger
This paper describes a method to directly fluorinate polyketides using a modified PKS enzyme, demonstrating its application in creating a fluorinated antibiotic derivative.
bioRxiv · Jul 30, 2021 · PreprintBiochemistry