Pharmacology & ToxicologyFrontiers in PharmacologyPeer-reviewed
A universal cannabinoid CB1 and CB2 receptor TR-FRET kinetic ligand binding assay.
Leire Borrega Roman, Bradley L. Hoare, Miroslav Kosar…·Dmitry B. Veprintsev
This paper develops a TR-FRET-based assay to measure ligand binding kinetics for CB1R and CB2R, finding that D77 enables accurate determination of on- and off-rates for various agonists and antagonists.
5 citations