Receptor levels determine binding affinity of WNT-3A to Frizzled 7 in a colorectal cancer model
L. Graetz, J. J. Sajkowska-Kozielewicz, J. Wesslowski, K. Petzold, G. Davidson, G. Schulte, P. Kozielewicz
The paper assesses WNT-3A binding affinity to endogenous versus overexpressed FZD7 in colorectal cancer cells and finds lower affinity with higher receptor concentrations.
bioRxiv · Jul 4, 2022Pharmacology & Toxicology