BiochemistryScience AdvancesPeer-reviewed
Structure-based discovery of highly bioavailable, covalent, broad-spectrum coronavirus-MPro inhibitors with potent in vivo efficacy
Tyler C. Detomasi, Gilles Degotte, Sijie Huang…·Charles S. Craik
This paper describes the discovery of new coronavirus MPro inhibitors with improved pharmacokinetics, broad-spectrum antiviral activity, and superior in vivo efficacy compared to existing drugs.
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