Pharmacology & ToxicologyProceedings of the National Academy of SciencesPeer-reviewed
Prolonged signaling of backbone-modified glucagon-like peptide-1 analogues with diverse receptor trafficking
Brian P. Cary, Marlies V. Hager, Zamara Mariam…·Samuel H. Gellman
This study identifies GLP-1 analogues with prolonged signaling by modifying specific amino acids, showing how receptor trafficking and peptide structure affect signaling duration.
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