Pharmacology & ToxicologybioRxivPreprint
Discovery of a pathway-selective platelet P2Y1R inverse agonist that suppresses inflammation while preserving hemostasis
Simon C. Pitchford, Kazi Sumaita Nahar, Dingxin Pan…·Khondaker Miraz Rahman
This paper designs a pathway-selective P2Y1R inverse agonist that suppresses inflammation without affecting hemostasis, demonstrating its functional selectivity in vitro and in vivo.
DOI 10.64898/2026.06.19.732319