Pharmacology & ToxicologybioRxivPreprint
Quinazoline-quinoline bisubstrate inhibitors target eukaryotic translation initiation factor 3 in Plasmodium falciparum
I. Dobrescu, E. Hammam, J. M. Dziekan…·F. Nardella
This study identifies PfEIF3i as a target of quinoline-quinazoline inhibitors in Plasmodium falciparum, showing its essential role in parasite development and potential as an antimalarial drug target.
DOI 10.1101/2022.12.10.519887