Pharmacology & ToxicologybioRxiv
Modifications in the piperazine ring of nucleozin affects anti-influenza activity
E. Correa-Padilla, A. Hernandez-Cano, G. Cuevas…·K. Martinez-Mayorga
The paper evaluates nucleozin analogs with modified piperazine rings, finding that increased conformational flexibility reduces anti-influenza activity and supports a QSAR model for predicting activity.
DOI 10.1371/journal.pone.0277073