BiochemistrybioRxiv
Diversity-oriented synthesis encoded by deoxyoligonucleotides
L. Hudson, J. W. Mason, M. V. Westphal…·K. Briner
The paper describes the design, synthesis, and validation of a 3.7 million-member DNA-encoded library using diversity-oriented synthesis to enhance structural diversity for drug discovery.
DOI 10.1038/s41467-023-40575-5