Cancer BiologybioRxiv
Target-driven design of a coumarinyl chalcone scaffold based novel EF2 Kinase inhibitor suppresses breast cancer growth in vivo
F. Comert Onder, N. Kahraman, E. Bellur Atici…·B. Ozpolat
The paper designs a coumarinyl chalcone scaffold-based inhibitor of eEF-2K, showing in vitro and in vivo efficacy against breast cancer.
DOI 10.1021/acsptsci.1c00030