BiochemistrybioRxivPreprint
A time-resolved Forster resonance energy transfer assay to investigate inhibitor binding to ABCG2
J. I. Mitchell-White, D. A. Briggs, S. J. Mistry…·I. D. Kerr
The paper introduces a TR-FRET assay to measure inhibitor binding to ABCG2 and confirms NBD dimerization correlates with a shift in inhibitor affinity.
DOI 10.1101/2023.10.27.564323