Cell BiologybioRxiv
A new chemotype of chemically tractable nonsteroidal estrogens based on a thienopyrimidine core.
V. R. Sammeta, J. D. Norris, S. Artham…·T. M. Willson
The paper identifies a new chemotype of nonsteroidal estrogens based on a thienopyrimidine core through targeted screening and structure-guided optimization.
DOI 10.1021/acsmedchemlett.2c00180