Pharmacology & ToxicologyJournal of Medicinal ChemistryPeer-reviewed
Three nitrogen atoms turn old kinase inhibitors into new targetable remedy
Balázs Besztercei, Réka Antal, Leena Tähtivaara…·Krisztián A. Kovács
This paper introduces photoactivatable VEGFR2 inhibitors that enhance retinal disease treatment by light-triggered activation, reducing required doses and systemic exposure.
DOI 10.1021/acs.jmedchem.6c01380