BiochemistrybioRxivPreprint
Cellular uptake of folate-olaparib conjugates via folate receptor-mediated endocytosis: Potential for selective delivery of DNA damage response inhibitors into tumour cells
Vassilios Bavetsias, Lisa Pickard, Sara Díaz-Sánchez…·Udai Banerji
This paper develops folate-olaparib conjugates that selectively enter FR-overexpressing tumor cells via endocytosis and inhibit PARylation.
DOI 10.64898/2026.09.23.752340