Identification, Characterization and Synthesis of Natural Parasitic Cysteine Protease Inhibitors -- More Potent Falcitidin Analogs
S. Brinkmann, S. Semmler, C. Kersten, M. A. Patras, M. Kurz, N. Fuchs, S. J. Hammerschmidt, J. Legac, P. E. Hammann, A. Vilcinskas, P. J. Rosenthal, T. Schirmeister, A. Bauer, T. F. Schaeberle
The paper identifies and synthesizes natural falcitidin analogs with enhanced inhibitory activity against parasitic cysteine proteases.
bioRxiv · Oct 30, 2021 · PreprintMicrobiology