Cancer BiologybioRxivPreprint
Small Molecule Inhibitors of the Human Histone Lysine Methyltransferase NSD2 / WHSC1 / MMSET Identified from a Quantitative High-Throughput Screen with Nucleosome Substrate
Nathan P. Coussens, Stephen C. Kales, Mark J. Henderson…·Matthew D. Hall
This study identifies five small molecule inhibitors of NSD2 through high-throughput screening and validates their activity in cell-based assays.
DOI 10.1101/208439