BiochemistryNature CommunicationsPeer-reviewed
Reinstating targeted protein degradation with DCAF1 PROTACs in CRBN PROTAC resistant settings
Martin Schröder, Martin Renatus, Xiaoyou Liang…·Claudio R. Thoma
This study develops DCAF1-based PROTACs to overcome CRBN resistance in targeted protein degradation, demonstrating effective degradation of BTK in CRBN-resistant cells.
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