BiophysicsJournal of Biological ChemistryPeer-reviewed
Structural determinants of the direct inhibition of GIRK channels by Sigma-1 receptor antagonist
Chang Liu, I‐Shan Chen, Michihiro Tateyama, Yoshihiro Kubo
This study identifies BD1047 as a direct inhibitor of GIRK channels, showing stronger inhibition of GIRK4 than GIRK2 and revealing structural determinants involving Leu77 on GIRK4.
5 citations