Cancer BiologybioRxiv
Epigenetic anti-cancer treatment with a stabilized carbocyclic Decitabine analogue
F. R. Traube, N. F. Bras, W. P. Roos…·T. Carell
This paper evaluates a stabilized carbocyclic Decitabine analogue, showing it effectively inhibits DNMT1 and induces more DNA damage in cancer cells with less toxicity.
DOI 10.1002/chem.202200640