MicrobiologybioRxiv
DNA-dependent binding of nargenicin to DnaE1 inhibits replication in Mycobacterium tuberculosis
M. D. Chengalroyen, M. K. Mason, A. Borsellini…·V. Mizrahi
This study shows nargenicin binds to Mtb DnaE1 DNA-dependent polymerase, inhibiting replication and inducing DNA damage response in tuberculosis bacteria.
DOI 10.1021/acsinfecdis.1c00643