A novel dimeric FAP-targeting small molecule-radio conjugate with high and prolonged tumour uptake
A. Galbiati, A. Zana, M. Bocci, J. Millul, A. Elsayed, J. Mock, D. Neri, S. Cazzamalli
This paper develops a dimeric FAP-targeting radioligand with prolonged tumour uptake and improved tumour-to-organ ratio, showing potent anti-tumour efficacy in preclinical models.
bioRxiv · Feb 21, 2022Pharmacology & Toxicology