Pharmacology & ToxicologybioRxivPreprint
Discovery of the first selective M4 muscarinic acetylcholine receptor antagonists with in vivo anti-parkinsonian and anti-dystonic efficacy
M. S. Moehle, A. M. Bender, J. W. Dickerson…·J. M. Rook
This paper discovers the first selective M4 muscarinic acetylcholine receptor antagonists and confirms their anti-parkinsonian and anti-dystonic efficacy in rodent models.
DOI 10.1101/2020.10.12.324152