BiochemistrybioRxiv
Dual-Probe Activity-Based Protein Profiling Reveals Site-Specific Differences in Protein Binding of EGFR-Directed Drugs
Wouter van Bergen, Kristina Žuna, Jan Fiala…·Marc P. Baggelaar
This study compares two EGFR-targeted drugs using ABPP to reveal site-specific binding differences and off-target effects at low concentrations.
DOI 10.1021/acschembio.3c00637