Pharmacology & ToxicologybioRxivPreprint
A small-molecule myosin inhibitor as a targeted multi-stage antimalarial
D. V. Trivedi, A. Karabina, G. Bergnes…·J. Spudich
This paper develops a small-molecule myosin inhibitor, KNX-115, effective against multiple stages of Plasmodium infection with high selectivity and potency.
DOI 10.1101/2022.09.09.507317