Pharmacology & ToxicologybioRxiv
Pharmacological Characterisation of Novel Adenosine Receptor A3R Antagonists
K. Barkan, P. Lagarias, M. Stampelou…·G. Ladds
This study characterizes a selective A3R antagonist, K18, and identifies its binding mode through molecular dynamics simulations and mutagenesis.
DOI 10.1038/s41598-020-74521-y