Cancer BiologybioRxiv
Protein mimetic amyloid inhibitor potently abrogates cancer-associated mutant p53 aggregation and restores tumor suppressor function
L. Palanikumar, L. Karpauskaite, S. Hassan…·M. Magzoub
This study identifies a small-molecule amyloid inhibitor that disrupts mutant p53 aggregation, restores its function, and reduces tumor growth in xenograft models.
DOI 10.1038/s41467-021-23985-1