Pharmacology & ToxicologybioRxivPreprint
ent-Verticilide B1 inhibits type 2 ryanodine receptor channels and is antiarrhythmic in Casq2-/- mice
A. Gochman, T. Q. Do, K. Kim…·B. C. Knollmann
This paper identifies ent-verticilide B1 as an antiarrhythmic compound that inhibits RyR2 channels and reduces arrhythmias in Casq2-/- mice.
DOI 10.1101/2023.07.03.547578