Pharmacology & ToxicologybioRxivPreprint
CGRP-receptor family reveals endogenous GPCR agonist bias and its significance in primary human cardiovascular cells
A. Clark, N. Mullooly, D. Safitri…·G. Ladds
The paper demonstrates endogenous agonist bias at the calcitonin-like receptor in primary human cardiovascular cells, showing physiological consequences through RAMP switching.
DOI 10.1101/2020.12.21.423730