Pharmacology & ToxicologyJournal of Medicinal ChemistryPeer-reviewed
Synthesis and Biological Evaluation of Nipecotic Acid Derivatives with Terminally Double-Substituted Allenic Spacers as mGAT4 Inhibitors
Maren Jung, Kinga Sałat, Georg C. Höfner…·Klaus T. Wanner
This paper synthesizes and evaluates nipecotic acid derivatives with allenic spacers as mGAT4 inhibitors, identifying a potent compound with anticonvulsant and anxiolytic effects in mice.
3 citations