Pharmacology & ToxicologybioRxivPreprint
Structure-Functional-Selectivity Relationship Studies on A-86929 Analogs and Small biaryl Fragments toward Discovery of biased D1 agonists
H. Li, R. Mirabel, J. Zimmerman…·N. M. Urs
This paper identifies chemical motifs for β-arrestin-biased D1R agonists through SAR studies of A-86929 analogs and small biaryl fragments.
DOI 10.1101/2021.10.01.462758