ImmunologybioRxivPreprint
Discovery of D2469079A, A novel selective Toll-Like Receptor 7/8 Antagonist with Brain Penetrance
Xiaobing Deng, Xun Zhang, Wenjia Tian…·Yijun Zhou
This paper identifies and characterizes D2469079A, a novel TLR7/8 antagonist with brain penetration, showing efficacy and safety in preclinical models.