BiochemistryBioorganic ChemistryPeer-reviewed
In Vitro Safety Signals for Potential Clinical Development of the Anti-Inflammatory Pregnane X Receptor Agonist FKK6
Zdeněk Dvořák, Barbora Vyhlídalová, Petra Pečinková…·Sridhar Mani
This paper performs in vitro pharmacological profiling of FKK6, showing high PXR selectivity, intestinal permeability, and rapid metabolism, supporting its potential preclinical development.
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