BiochemistryEuropean Journal of Medicinal ChemistryPeer-reviewed
Substitutions at the C-8 position of quinazolin-4-ones improve the potency of nicotinamide site binding tankyrase inhibitors
Chiara Bosetti, Dionysis Kampasis, Shoshy Alam Brinch…·Ioannis K. Kostakis
This study identifies C-8 position substitutions in quinazolin-4-ones that enhance the potency and selectivity of tankyrase inhibitors by improving interactions with TNKS2.
5 citations