Pharmacology & ToxicologyBioorganic & Medicinal ChemistryPeer-reviewed
Identification and Characterization of the First Fragment Hits for SETDB1 Tudor Domain
P. Mader, R. Mendoza-Sanchez, A. Iqbal…·C. Arrowsmith
The paper identifies small molecule fragments that bind to the tudor domain of SETDB1 and describes their binding modes and biophysical properties.
DOI 10.1016/j.bmc.2019.07.020