BiochemistrybioRxiv
Comparative analysis of drug-like EP300/CREBBP acetyltransferase inhibitors
M. C. Crawford, D. R. Tripu, S. A. Barritt…·J. L. Meier
This study compares the biochemical and biological potencies of three EP300/CREBBP acetyltransferase inhibitors and demonstrates their utility in investigating epigenetic mechanisms.
DOI 10.1021/acschembio.3c00293