BiochemistrybioRxiv
PKD autoinhibition in trans regulates activation loop autophosphorylation in cis
R. Reinhardt, K. Hirzel, G. Link…·T. A. Leonard
This study shows PKD is regulated by trans-autoinhibition followed by cis autophosphorylation, switching the kinase on by preventing re-autoinhibition.
DOI 10.1073/pnas.2212909120